Bayer receives MHRA authorisation for new indication of Nubeqa® (darolutamide) plus androgen deprivation therapy as a treatment option in metastatic hormone-sensitive prostate cancer

  • The marketing authorisation is based on results from the pivotal Phase III ARANOTE trial evaluating the efficacy and safety of darolutamide, an oral androgen receptor inhibitor, plus androgen deprivation therapy (ADT) in adult patients with metastatic hormone-sensitive prostate cancer (mHSPC)1 

  • In the UK, prostate cancer is the most common cancer in men, with over 55,000 men getting diagnosed each year and more than 15,000 new cases confirmed as metastatic prostate cancer.2,3  

  • Darolutamide plus ADT is now licensed in the UK for use as a treatment option in mHSPC, with and without chemotherapy docetaxel,1 based on two pivotal Phase III studies in mHSPC4,5 

The UK’s Medicines and Healthcare products Regulatory Agency (MHRA) has authorised the use of Nubeqa® (darolutamide) for the treatment of adult patients with metastatic hormone-sensitive prostate cancer (mHSPC) in combination with androgen deprivation therapy (ADT).1  

 

The authorisation is based on positive results from the pivotal Phase III ARANOTE trial, evaluating the efficacy and safety of darolutamide plus ADT in patients with mHSPC. The trial showed that darolutamide plus ADT significantly improved radiological progression-free survival (rPFS), reducing the risk of radiological progression or death by 46% (HR 0.54; 95% CI 0.41–0.71; P<0.0001), compared to placebo plus ADT.4 The rPFS rates at 24 months were 70.3% in the darolutamide group and 52.1% in the placebo group. Consistent benefits in rPFS were observed across prespecified subgroups, including in patients with high-volume (HR 0.60; 95% CI 0.44-0.80) and low-volume (HR 0.30; 95% CI 0.15-0.60) mHSPC.4 The incidence of treatment-emergent adverse events (TEAEs) was similar between treatment groups.4 Treatment discontinuations due to TEAEs were lower in patients receiving darolutamide plus ADT compared to placebo plus ADT (6.1% vs 9.0%).4 

 

"Despite significant advances in prostate cancer care, there is still a need for widening the options for men with advanced prostate cancer that can maintain quality of life as much as possible alongside improving their outcomes from prostate cancer, meaning more quality time overall. This means we have to adapt treatment to the individual person, taking into account other medical problems, such as medication, age and what their treatment goals and preferences are,” said Professor Alison Birtle, Consultant Clinical Oncologist at the Rosemere Cancer Centre, Lancashire Teaching Hospitals, Honorary Clinical Professor in the Faculty of Biology, Medicine & Health at the University of Manchester and Honorary Clinical Professor at The University of Central Lancashire. “Today’s authorisation of darolutamide plus ADT for use in metastatic hormone-sensitive prostate cancer provides me and other UK physicians with greater flexibility to tailor treatment to an individual patient's needs.” 

 

“The authorisation represents an important development in treatment options for people living with metastatic hormone-sensitive prostate cancer in the UK. Our focus now is to ensure this new treatment option is available to patients and physicians as quickly as possible,” said Dr. Joep Hufman, Country Medical Director, Bayer UK & Ireland. “We remain committed to advancing treatment options for patients that address unmet needs across all stages of disease, which may help delay disease progression while maintaining quality of life.”  

 

In the UK, prostate cancer is the most common cancer in men, with over 55,000 new cases identified each year.2 It accounts for nearly 28% of all new cancer diagnoses (2017 – 2019),2 highlighting the significant impact of this disease on public health. There are around 12,000 prostate cancer deaths in the UK every year – that’s 33 men every day (2017 – 2019), making it the second leading cause of cancer-related deaths in the country.2 The incidence of prostate cancer is expected to continue to rise by

15% in the UK2 due to an aging population and improved screening practices.6 While early-stage prostate cancer has a high survival rate, the challenges associated with advanced disease underscore the need for continued research and the development of future treatment options.7 

 

“Advanced prostate cancer presents profound challenges that significantly affect not only patients but also their families. The emotional and psychological toll of a diagnosis of metastatic prostate cancer adds another layer of difficulty, often resulting in anxiety and distress. It is crucial that we continue to raise awareness and advocate for better access to timely diagnosis, effective treatments, and comprehensive support services that the patients and their families need to navigate this challenging journey,” said Oliver Kemp, CEO, Prostate Cancer Research. 

 

Darolutamide was authorised in March 2020 in the European Union under the brand name Nubeqa® for the treatment of adult men with non-metastatic castration resistant prostate cancer (nmCRPC), who are at high risk of developing metastatic disease.8 It was authorised in November 2022 in the UK for the treatment of adult patients with mHSPC in combination with ADT and docetaxel.9 In May 2023, the National Institute for Health and Care Excellence (NICE) issued guidance (TA903) recommending darolutamide plus ADT in combination with docetaxel as a treatment option for patients with mHSPC.10  

 

ENDS 

Bayer Media Contact : 

Veronica Yao, +44 (0) 7870 485 926 

 

Notes to Editors 

About metastatic hormone-sensitive prostate cancer (mHSPC) 

mHSPC is cancer that has spread beyond the prostate to other parts of the body but still responds to treatment with hormone therapy.11 mHSPC precedes the development of metastatic castration-resistant prostate cancer (mCRPC),12 which no longer responds to treatment with hormone therapy. 

Despite treatment, most men with mHSPC will eventually progress to mCRPC,13 a condition with limited survival. 

 

About the ARANOTE Trial 

The ARANOTE trial is a randomised, double-blind, placebo-controlled Phase III study designed to assess the efficacy and safety of darolutamide plus androgen deprivation therapy (ADT) in patients with metastatic hormone-sensitive prostate cancer (mHSPC). 669 patients were randomised 2:1 to receive either 600mg of darolutamide twice daily or placebo in addition to ADT.14 

 

The primary endpoint of this study was radiological progression-free survival (rPFS), measured as time from randomisation to date of first documented radiological progressive disease or death due to any cause, whichever occurs first. Secondary endpoints include overall survival (time to death from any cause), time to CRPC (castration-resistant prostate cancer) event, time to initiation of subsequent anti-cancer therapy, time to prostate-specific antigen (PSA) progression, PSA undetectable rates, time to pain progression, and safety assessments.14 

 

About prostate cancer at Bayer  

Bayer is committed to delivering science for a better life by advancing a portfolio of innovative treatments. The company has the passion and determination to develop new medicines that help improve and extend the lives of people living with cancer. Prostate cancer is the second most commonly diagnosed cancer in men globally (based on data from 2020)15, the most common cancer in men in the UK, and a key area of focus for Bayer. Bayer is focused on addressing the unique needs of patients with prostate cancer, providing treatments that could potentially extend their lives throughout the different stages of the disease and allowing them to continue with their everyday activities so that patients can live longer and better lives. 

 

About Bayer  

Bayer is a global enterprise with core competencies in the life science fields of health care and nutrition. In line with its mission, “Health for all, Hunger for none,” the company’s products and services are designed to help people and the planet thrive by supporting efforts to master the major challenges presented by a growing and aging global population. Bayer is committed to driving sustainable development and generating a positive impact with its businesses. At the same time, the Group aims to increase its earning power and create value through innovation and growth. The Bayer brand stands for trust, reliability and quality throughout the world. In fiscal 2024, the Group employed around 93,000 people and had sales of 46.6 billion euros. R&D expenses amounted to 6.2 billion euros. For more information, go to www.bayer.co.uk. 

 

Forward-Looking Statements  

This release may contain forward-looking statements based on current assumptions and forecasts made by Bayer management. Various known and unknown risks, uncertainties and other factors could lead to material differences between the actual future results, financial situation, development or performance of the company and the estimates given here. These factors include those discussed in Bayer’s public reports which are available on the Bayer website at www.bayer.co.uk. The company assumes no liability whatsoever to update these forward-looking statements or to conform them to future events or developments.  

 

 

References 

  1. Summary of Product Characteristics (SmPC) for Nubeqa 300 mg film-coated tablets.  

  2. Cancer Research UK. Prostate cancer statistics. Available at: https://www.cancerresearchuk.org/health-professional/cancer-statistics/statistics-by-cancer-type/prostate-cancer. Last accessed: May 2025. 

  3. Prostate Cancer UK. Advanced prostate cancer: your questions answered about the disease affecting Bill Turnbull. Available at: https://prostatecanceruk.org/about-us/news-and-views/2018/10/advanced-disease-blog.  Last accessed: May 2025. 

  4. Saad F. et al. Darolutamide in Combination With Androgen-Deprivation Therapy in Patients With Metastatic Hormone-Sensitive Prostate Cancer From the Phase III ARANOTE Trial. doi/10.1200/JCO September 2024. Available at: https://ascopubs.org/doi/10.1200/JCO-24-01798  

  5. Smith, RA, et al. Darolutamide and Survival in Metastatic, Hormone-Sensitive Prostate Cancer. doi:/10.1056/NEJMoa2119115. Published on February 17, 2022, at NEJM.org.  

  6. Schafer EJ, et al. The incidence of prostate cancer is expected to continue to rise due to an aging population and improved screening practices. European Urology. Volume 87, Issue 3, March 2025, Pages 302-313. https://doi.org/10.1016/j.eururo.2024.11.013  

  7. The future of prostate cancer research: what could the next decade bring? The Institute of Cancer Research. Available at: https://www.icr.ac.uk/about-us/icr-news. Last accessed: May 2025. 

  8. Nubeqa (darolutamide). European Medicines Agency. Available from:  https://www.ema.europa.eu/en/medicines/human/EPAR/nubeqa#authorisation-details-section Last accessed: May 2025. 

  9. NUBEQA® (darolutamide) 300 mg film-coated tables Summary of Product Characteristics. Available at: https://www.medicines.org.uk/emc/product/11324 Last accessed: May 2025.  

  10. Final draft guidance. National Institute for Health and Care Excellence. Darolutamide with androgen deprivation therapy and docetaxel for treating hormone-sensitive metastatic prostate cancer. Available from: https://www.nice.org.uk/guidance/gid-ta10860/documents/final-appraisal-determination-document Last accessed: May 2025. 

  11. Cancer.Net. ASCO answers: Prostate Cancer. Available at: https://www.cancer.net/sites/cancer.net/files/asco_answers_guide_prostate.pdf Last accessed: April 2025. 

  12. Cattrini, et al. Current Treatment Options for Metastatic Hormone-Sensitive Prostate Cancer. Cancers.2019 11(9), p.1355 

  13. Ritch, C. and Cookson, M. Recent trends in the management of advanced prostate cancer. F1000Res. 2018 Sep 21;7:F1000 Faculty Rev-1513. 

  14. Darolutamide in Addition to ADT Versus ADT in Metastatic Hormone-sensitive Prostate Cancer (ARANOTE). Clinicaltrial.gov. Available at: https://www.clinicaltrials.gov/study/NCT04736199. Last accessed: May 2025. 

  15. Bray F et al. Global cancer statistics 2022: GLOBOCAN estimates of incidence and mortality worldwide for 36 cancers in 185 countries. https://acsjournals.onlinelibrary.wiley.com/doi/10.3322/caac.21834. Last accessed: May 2025.  

 

 

RP-NUB-GB-0783 / May 2025